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Chemical Name:Tamoxifen citrateSynonymsNOLVADEX;TMX;tamoxifene;SoltaMox;Nolvadex(Tamoxifen);(Z)-[2-[4-(1,2-diphenylbut-1-enyl)phenoxy]ethyl]dimethylammonium dihydrogen 2-hydroxypropane-1,2,3-tricarboxylate;TMX1;TXNDC;Adopan;kessarCBNumber:CB7853805Molecular Formula:C32H37NO8Molecular Weight:563.64Melting point 140-144 °Cstorage temp. 2-8°Csolubility methanol: soluble50mg/mL, clear, colorlessform Powdercolor White to off-whiteWater Solubility slightly solubleSensitive Light Sensitive & HygroscopicUsesTamoxifen citrate is commonly used in the treatment of women with metastatic carcinoma of the breast to prevent recurrence after surgery or radiation treatment, and as prophylaxis for patients at very high risk to develop breast cancer.Usesanti-estrogen, protein kinase C inhibitor, beneficial cardiovascular effects, bone cancer treatment, induces DNA adduct formationUsesTamoxifen Citrate is a selective estrogen response modifier (SERM), protein kinase C inhibitor and anti-angiogenetic factor. Tamoxifen is a prodrug that is metabolized to active metabolites 4-hydroxytamoxifen (4-OHT) and endoxifen by cytochrome P450 isoforms CYP2D6 and CYP3A4. 

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